Publications
Alex N. Eberle has published two books and edited various conference proceedings, and he is an author or coauthor of more than 200 articles. The links to the publications are password-protected; please contact the author if you are interested in a specific paper.
Books
Schneider CH, Eberle AN (eds). Peptides 1992; Proceedings of the 22nd European Peptide Symposium. Escom 1993.
Vaudry H, Eberle AN (eds). The Melanotropic Peptides. NY Acad Sci 1993; 680: i-xvi and 1-687.
Eberle AN. The Melanotropins: Chemistry, Physiology and Mechanisms of Action. Karger 1988.
Eberle AN, Geiger R, Wieland T (eds.). Perspectives in Peptide Chemistry. Karger 1981.
Skoda R, Eberle AN (eds.). Department of Research; a Portrait 1978-2005. Morf, Basel 2005.
2013
2012
2011
2010
- Eberle AN, Mild G, Zumsteg U. Cellular models for the study of the pharmacology and signaling of melanin-concentrating hormone receptors. J Recept Signal Transduct 2010; 30(6):385-402.
- Mastofrancesco A, Kokot A, Eberle AN, Gibbons NCJ, Schallreuter KU, Strozyk E, Picardo M, Zouboulis CC, Luger TA, Böhm M. KDPT, a tripeptide derivative of alpha-melanocyte-stimulating hormone, suppresses IL-1beta-mediated cytokine expression and signaling in human sebocytes. J Immunol 2010; 185:1903-1911.
- Eberle AN, Bapst J-P, Calame M, Tanner H, Froidevaux S. MSH radiopeptides for targeting melanoma metastases. In: Advances in Experimental Medicine and Biology, Vol 681, Melanocortins: Multiple Actions and Therapeutic Potential, A. Catania (ed.), 133-142, Springer Science+Business Media, Landes Bioscience (2010).
- Lindinger A, Peterli R, Peters T, Kern B, von Flüe M, Calame M, Hoch M, Eberle AN, Lindinger PW. Mitochondrial DNA content in human omental adipose tissue. Obes Surg 2010;20(1):84-92.
2009
- Eberle AN. Targeting of melanoma metastases with peptides. Pigment Cell Melanoma Res 2009; 22: 655-656.
- Eberle AN, Mild G. Receptor-mediated tumor targeting with radiopeptides. Part 1. General principles and methods. J Recept Signal Transduct Res 2009;29(1):1-37.
- Bapst JP, Calame M, Tanner H, Eberle AN. Glycosylated DOTA-α-Melanocyte-Stimulating Hormone Analogues for Melanoma Targeting: Influence of the Site of Glycosylation on in Vivo Biodistribution. Bioconjug Chem 2009;20:984-993.
- Knecht S, Ricklin D, Eberle AN, Ernst B. Oligohis-tags: mechanisms of binding to Ni2+-NTA surfaces. J Mol Recognit 2009;22(4):270-279.
2008
- Hoch M, Hirzel E, Lindinger P, Eberle AN, Linscheid P, Martin I, Peters T, Peterli R. Weak functional coupling of the melanocortin-1 receptor expressed in human adipocytes. J Recept Signal Transduct Res 2008;28(5):485-504.
- Hoch M, Eberle AN, Peterli R, Peters T, Seboek D, Keller U, Muller B, Linscheid P. LPS induces interleukin-6 and interleukin-8 but not tumor necrosis factor-alpha in human adipocytes. Cytokine 2008;41(1):29-37.
2007
- Bapst JP, Froidevaux S, Calame M, Tanner H, Eberle AN. Dimeric DOTA-alpha-melanocyte-stimulating hormone analogs: synthesis and in vivo characteristics of radiopeptides with high in vitro activity. J Recept Signal Transduct Res 2007;27(5-6):383-409.
- Hoch M, Eberle AN, Wagner U, Bussmann C, Peters T, Peterli R. Expression and localization of melanocortin-1 receptor in human adipose tissues of severely obese patients. Obesity (Silver Spring) 2007;15(1):40-49.
2006
- Peterli R, Peters T, von Flüe M, Hoch M, Eberle AN. Melanocortin-4 receptor gene and complications after gastric banding. Obes Surg 2006;16(2):189-195.
- Jégou S, Cone RD, Eberle AN, Vaudry H. Melanocortins. In: Handbook of biologically active peptides, A. Kastin (ed.), 96:689-696, Elsevier/Academic Press (2006).
2005
- Eberle AN, Beglinger C. Does 177Lu-labeled octreotate improve the rate of remission of endocrine gastroenteropancreatic tumors? Nat Clin Pract Endocrinol Metab 2005;1(1):20-21.
- Szokolóczi O, Schwab R, Peták I, Orfi L, Pap A, Eberle AN, Szüts T, Kéril G. TT232, a novel signal transduction inhibitory compound in the therapy of cancer and inflammatory diseases. J Recept Signal Transduct Res 2005;25(4-6):217-235.
- Froidevaux S, Calame-Christe M, Tanner H, Eberle AN. Melanoma targeting with DOTA-alpha-melanocyte-stimulating hormone analogs: structural parameters affecting tumor uptake and kidney uptake. J Nucl Med 2005;46(5):887-895.
2004
- Eberle AN, Mild G, Froidevaux S. Receptor-mediated tumor targeting with radiopeptides. Part 1. General concepts and methods: applications to somatostatin receptor-expressing tumors. J Recept Signal Transduct Res 2004;24(4):319-455.
- Eberle AN, Mild G, Schlumberger S, Drozdz R, Hintermann E, Zumsteg U. Expression and characterization of melanin-concentrating hormone receptors on mammalian cell lines. Peptides 2004;25(10):1585-1595.
- Froidevaux S, Calame-Christe M, Schuhmacher J, Tanner H, Saffrich R, Henze M, Eberle AN. A gallium-labeled DOTA-alpha-melanocyte- stimulating hormone analog for PET imaging of melanoma metastases. J Nucl Med 2004;45(1):116-123.
- Eberle AN, Froidevaux S. Dota-chelator-containing radiopeptides for the targeting of tumour metastases. Act Chim Thér 2004;30:209-228.
- Froidevaux S, Calame M, Tanner H, Schumacher J, Eberle AN. Targeting of melanoma metastases with 111In/68Ga-DOTA-labeled analogs of alpha-melanocyte-stimulating hormone. 5th International Symposium on Regulatory Peptides. Abstract 43. Regul Pept 2004;122:16.
- Froidevaux S, Calame M. Tanner H, Schumacher J, Eberle AN. 41. Receptor-mediated targeting of melanoma metastases with a-MSH radio-peptides. In: Proc 8th Int Symp on Synthesis (Peptides, Proteins and Nucleic Acids), R. Epton (ed.), 183-186, Mayflower Worldwide (2004).
2003
- Eberle AN, Froidevaux S. Radiolabeled alpha-melanocyte-stimulating hormone analogs for receptor-mediated targeting of melanoma: from tritium to indium. J Mol Recognit 2003;16(5):248-254.
- Froidevaux S, Calame-Christe M, Sumanovski L, Tanner H, Eberle AN. DOTA alpha-melanocyte-stimulating hormone analogues for imaging metastatic melanoma lesions. Ann N Y Acad Sci 2003;994:378-383.
- Schlumberger SE, Saito Y, Giller T, Hintermann E, Tanner H, Jäggin V, Zumsteg U, Civelli O, Eberle AN. Different structural requirements for melanin-concentrating hormone (MCH) interacting with rat MCH-R1 (SLC-1) and mouse B16 cell MCH-R. J Recept Signal Transduct Res 2003;23(1):69-81.
- Eberle AN, Zumsteg U, Jäggin V, Bódi J, Orosz G, Süli-Vargha H. Agouti protein: pleiotropic functions and mechanisms of action. 3rd Hellenic Forum on Bioactive Peptides, 155-166 (2003).
2002
- Schlumberger SE, Talke-Messerer C, Zumsteg U, Eberle AN. Expression of receptors for melanin-concentrating hormone (MCH) in different tissues and cell lines. J Recept Signal Transduct Res 2002;22(1-4):509-531.
- Froidevaux S, Eberle AN. Homologous regulation of melanocortin-1 receptor (MC1R) expression in melanoma tumor cells in vivo. J Recept Signal Transduct Res 2002;22(1-4):111-121.
- Froidevaux S, Calame-Christe M, Tanner H, Sumanovski L, Eberle AN. A novel DOTA-alpha-melanocyte-stimulating hormone analog for metastatic melanoma diagnosis. J Nucl Med 2002;43(12):1699-1706.
- Wunderlich K, Golubnitschaja O, Pache M, Eberle AN, Flammer J. Increased plasma levels of 20S proteasome alpha-subunit in glaucoma patients: an observational pilot study. Mol Vis 2002;8:431-435.
- Froidevaux S, Eberle AN. Somatostatin analogs and radiopeptides in cancer therapy. Biopolymers 2002;66(3):161-183.
- Schlumberger SE, Jäggin V, Tanner H, Eberle AN. Endogenous receptor for melanin-concentrating hormone in human neuroblastoma Kelly cells. Biochem Biophys Res Commun 2002;298(1):54-59.
- Huwyler J, Cerletti A, Fricker G, Eberle AN, Drewe J. By-passing of P-glycoprotein using immunoliposomes. J Drug Target 2002;10(1):73-79.
- Froidevaux S, Eberle AN, Christe M, Sumanovski L, Heppeler A, Schmitt JS, Eisenwiener K, Beglinger C, Mäcke HR. Neuroendocrine tumor targeting: study of novel gallium-labeled somatostatin radiopeptides in a rat pancreatic tumor model. Int J Cancer 2002;98(6):930-937.
2001
- Hintermann E, Tanner H, Talke-Messerer C, Schlumberger S, Zumsteg U, Eberle AN. Interaction of melanin-concentrating hormone (MCH), neuropeptide E-I (NEI), neuropeptide G-E (NGE), and alpha-MSH with melanocortin and MCH receptors on mouse B16 melanoma cells. J Recept Signal Transduct Res 2001;21(1):93-116.
- Eberle AN, Bódi J, Orosz G, Süli-Vargha H, Jäggin V, Zumsteg U. Antagonist and agonist activities of the mouse agouti protein fragment (91-131) at the melanocortin-1 receptor. J Recept Signal Transduct Res 2001;21(1):25-45.
- Liu R, Hintermann E, Erb C, Tanner H, Flammer J, Eberle AN, Haefliger IO. Modulation of Na/K-ATPase activity by isoproterenol and propranolol in human non-pigmented ciliary epithelial cells. Klin Monatsbl Augenheilkd 2001;218(5):363-365.
- Schwab RE, Froidevaux S, Paku S, Tejeda M, Szende B, Pap A, Beglinger C, Eberle AN, Kéri G. Antiproliferative efficacy of the somatostatin analogue TT-232 in human melanoma cells and tumours. Anticancer Res 2001;21(1A):71-75.
- Hintermann E, Erb C, Talke-Messerer C, Liu R, Tanner H, Flammer J, Eberle AN. Expression of the melanin-concentrating hormone receptor in porcine and human ciliary epithelial cells. Invest Ophthalmol Vis Sci 2001;42(1):206-209.
- Froidevaux S, Meier A-M, Heppeler A, Mäcke HR, Beglinger C, Eberle AN. 70. Radiolabelled DOTA-somatostatin analogues for tumour diagnosis and internal radiotherapy. In: Solid Phase Synthesis & Combinatorial Libraries 2000, R. Epton (ed.), 281-284, Mayflower, Kingswinford, U.K., 2001.
- Froidevaux S, Christe M, Heppeler A, Mäcke HR, Beglinger C, Eberle AN. Radioactive peptides for receptor-mediated targeting of tumours. 2nd Hellenic Forum on Bioactive Peptides, 155-164 (2001).
- Eberle AN, Bódi J, Orosz G, Süli-Vargha H, Jäggin V, Zumsteg U. In: Peptides: The Wave of the Future. Lebl M, Houghton RA (eds.), 1-2, American Peptide Society 2001.
2000
- Cerletti A, Drewe J, Fricker G, Eberle AN, Huwyler J. Endocytosis and transcytosis of an immunoliposome-based brain drug delivery system. J Drug Target 2000;8(6):435-446.
- Wunderlich K, Pech M, Eberle AN, Mihatsch M, Flammer J, Meyer P. Expression of connective tissue growth factor (CTGF) mRNA in plaques of human anterior subcapsular cataracts and membranes of posterior capsule opacification. Curr Eye Res 2000;21(2):627-636.
- Froidevaux S, Heppeler A, Eberle AN, Meier AM, Häusler M, Beglinger C, Béhé M, Powell P, Mäcke HR. Preclinical comparison in AR4-2J tumor-bearing mice of four radiolabeled 1,4,7,10-tetraazacyclododecane-1,4,7,10-tetraacetic acid-somatostatin analogs for tumor diagnosis and internal radiotherapy. Endocrinology 2000;141(9):3304-3312.
- Heppeler A, Froidevaux S, Eberle AN, Maecke HR. Receptor targeting for tumor localisation and therapy with radiopeptides. Curr Med Chem 2000;7(9):971-994.
- Bigliardi-Qi M, Bigliardi PL, Eberle AN, Büchner S, Rufli T. beta-endorphin stimulates cytokeratin 16 expression and downregulates mu-opiate receptor expression in human epidermis. J Invest Dermatol 2000;114(3):527-532.
- Eberle AN, Froidevaux S, Siegrist W. 17. Melanocortins and melanoma. In: The Melanocortin Receptors (R. Cone, ed.), 491-520 (2000), Humana Press Inc., Totowa, NJ.
- Eberle AN. 1. Proopiomelanocortin and the melanocortin peptides. In: The Melanocortin Receptors (R. Cone, ed.), 3-67 (2000), Humana Press Inc., Totowa, NJ.
1999
- Froidevaux S, Hintermann E, Török M, Mäcke HR, Beglinger C, Eberle AN. Differential regulation of somatostatin receptor type 2 (sst 2) expression in AR4-2J tumor cells implanted into mice during octreotide treatment. Cancer Res 1999;59(15):3652-3657.
- Drozdz R, Hintermann E, Tanner H, Zumsteg U, Eberle AN. (D-(p-benzoylphenylalanine)13, tyrosine19)-melanin-concentrating hormone, a potent analogue for MCH receptor crosslinking. J Pept Sci 1999;5(5):234-242.
- Huwyler J, Froidevaux S, Roux F, Eberle AN. Characterization of transferring receptor in an immortalized cell line of rat brain endothelial cells, RBE4. J Recept Signal Transduct Res 1999;19(1-4):729-739.
- Brandenburger Y, Rose K, Bagutti C, Eberle AN. Synthesis and receptor binding analysis of thirteen oligomeric alpha-MSH analogs. J Recept Signal Transduct Res 1999;19(1-4):467-480.
- Heizmann G, Hildebrand P, Tanner H, Ketterer S, Pansky A, Froidevaux S, Beglinger C, Eberle AN. A combinatorial peptoid library for the identification of novel MSH and GRP/bombesin receptor ligands. J Recept Signal Transduct Res 1999;19(1-4):449-466.
- Hintermann E, Drozdz R, Tanner H, Eberle AN. Synthesis and characterization of new radioligands for the mammalian melanin-concentrating hormone (MCH) receptor. J Recept Signal Transduct Res 1999;19(1-4):411-422.
- Froidevaux S, Meier M, Häusler M, Mäcke H, Beglinger C, Eberle AN. A microplate binding assay for the somatostatin type-2 receptor (SSTR2). J Recept Signal Transduct Res 1999;19(1-4):167-180.
- Hintermann E, Drozdz R, Tanner H, Zumsteg U, Eberle AN. 76. Radioligands for the receptor of mammalian melanin-concentrating hormone (MCH). In: Peptide Science – Present and Future, Y. Shimonishi (ed.), 226-227, Kluwer Academic Publishers (1999).
- Froidevaux S, Heppeler A, Behe M, Jermann E, Otte A, Müller-Brand J, Mäcke HR, Hildebrand P, Beglinger C, Eberle AN. 226. Peptide radiopharmaceuticals: studies of somatostatin receptors and ligands for tumor targeting. In: Peptide Science – Present and Future, Y. Shimonishi (ed.), 670-673, Kluwer Academic Publishers (1999).
- Eberle AN, Froidevaux S, Meier M, Jäggin V, Bódi J, Orosz G, Süli-Vargha H. Synthetic agouti protein fragment (91-131) is an inverse agonist of the melanocortin-1 (MC-1) receptor. In: Peptides 1998, S. Bajusz, F Hudecz (eds.), Akadémiai Kiadó, Budapest (1999).
- Hintermann E, Drozdz R, Tanner H, Eberle AN. 44. Synthesis and receptor binding activity of analogues and fragments of human melanin-concentrating hormone (MCH). In: Innovation and Perspectives in Solid Phase Synthesis & Combinatorial Libraries 1998, R. Epton (ed.), 193-196, Mayflower Scientific Limited, Birmingham (1999).
- Heppeler A, Froidevaux S, Mäcke HR, Jermann E, Béhé M, Powell P, Henning M. Radiometal-Labelled Macrocyclic Chelator-Derivatised Somatostatin Analogue with Superb Tumour-Targeting Properties and Potential for Receptor-Mediated Internal Radiotherapy. Chem Eur J 1999;5(7):1947-1981.
1998
- Drozdz R, Hintermann E, Eberle AN. Characterization of the receptor for melanin-concentrating hormone on melanoma cells by photocrosslinking. Ann N Y Acad Sci 1998;839:210-213.
- Siegrist W, Hintermann E, Roggo CN, Apfel CM, Klaus M, Eberle AN. Melanoma cell growth inhibition and melanocortin receptor downregulation induced by selective and non-selective retinoids. Melanoma Res 1998;8(2):113-122.
- Vallarino M, Trabucchi M, Chartrel N, Jäggin V, Eberle AN, Vaudry H. Melanin-concentrating hormone system in the brain of the lungfish Protopterus annectens. J Comp Neurol 1998;390(1):41-51.
- Heizmann G, Hildebrand P, Tanner H, Ketterer S, Beglinger C, Eberle AN. 32. Peptoid and hybrid peptoid-peptide ligands for the MSH and the GRP-preffering bombesin receptor developed from a combinatorial peptoid library. In: Peptides 1996, R. Ramage, R. Epton (eds.), 161-164, The European Peptide Society (1998).
1997
- Chluba-de Tapia J, de Tapia M, Jäggin V, Eberle AN. Cloning of a human multispanning membrane protein cDNA: evidence for a new protein family. Gene 1997;197(1-2):195-204.
- Heizmann G, Eberle AN. Xanthines as a scaffold for molecular diversity. Mol Divers 1997;2(3):171-174.
- Innamorati G, Sadeghi H, Eberle AN, Birnbaumer M. Phosphorylation of the V2 vasopressin receptor. J Biol Chem 1997;272(4):2486-2492.
- Pansky A, Peng F, Eberhard M, Baselgia L, Siegrist W, Baumann JB, Eberle AN, Beglinger C, Hildebrand P. Identification of functional GRP-preferring bombesin receptors on human melanoma cells. Eur J Clin Invest 1997;27(1):69-76.
- Baumann JB, Bagutti C, Siegrist W, Christen E, Zumsteg U, Eberle AN. MSH receptors and the response of human A375 melanoma cells to interleukin-1 beta. J Recept Signal Transduct Res 1997;17(1-3):199-210.
- Siegrist W, Drozdz R, Cotti R, Willard DH, Wilkison WO, Eberle AN. Interactions of alpha-melanotropin and agouti on B16 melanoma cells: evidence for inverse agonism of agouti. J Recept Signal Transduct Res 1997;17(1-3):75-98.
- Heizmann G, Tanner H, Eberle AN. 83. New ligands for the human melanoma MSH receptor identified by a peptoid library (oligo N-substituted glycines). In: Innovation and Perspectives in Solid Phase Synthesis & Combinatorial Libraries 1996: Peptides, Proteins and Nucleic Acids, R. Epton (ed.), 391-394, Mayflower Scientific, Birmingham (1997).
1996
- Chluba-de Tapia J, Bagutti C, Cotti R, Eberle AN. Induction of constitutive melanogenesis in amelanotic mouse melanoma cells by transfection of the human melanocortin-1 receptor gene. J Cell Sci 1996;109(Pt 8):2023-2030.
- Lichtensteiger W, Hanimann B, Siegrist W, Eberle AN. Region- and stage-specific patterns of melanocortin receptor ontogeny in rat central nervous system, cranial nerve ganglia and sympathetic ganglia. Brain Res Dev Brain Res 1996;91(1):93-110.
- Siegrist W, Willard DH, Wilkison WO, Eberle AN. Agouti protein inhibits growth of B16 melanoma cells in vitro by acting through melanocortin receptors. Biochem Biophys Res Commun 1996;218(1):171-175.
1995
- Siegrist W, Eberle AN. Melanocortins and their implication in melanoma. Trends Endocrinol Metab 1995;6(4):115-120.
- Drozdz R, Siegrist W, Baker BI, Chluba-de Tapia J, Eberle AN. Melanin-concentrating hormone binding to mouse melanoma cells in vitro. FEBS Lett 1995;359(2-3):199-202.
- Drozdz R, Eberle AN. Synthesis and iodination of human (phenylalanine 13, tyrosine 19) melanin-concentrating hormone for radioreceptor assay. J Pept Sci 1995;1(1):58-65.
- Drozdz R, Eberle AN. Binding sites for melanin-concentrating hormone (MCH) in brain synaptosomes and membranes from peripheral tissues identified with highly tritiated MCH. J Recept Signal Transduct Res 1995;15(1-4):487-502.
- Bagutti C, Oestreicher M, Siegrist W, Oberholzer M, Eberle AN. alpha-MSH receptor autoradiography on mouse and human melanoma tissue sections and biopsies. J Recept Signal Transduct Res 1995;15(1-4):427-442.
- Siegrist W, Sauter P, Eberle AN. A selective protein kinase C inhibitor (CGP 41251) positively and negatively modulates melanoma cell MSH receptors. J Recept Signal Transduct Res 1995;15(1-4):283-296.
- Chluba-de Tapia J, Bagutti C, Wikberg JS, Chhajlani V, Eberle AN. Stable expression of the human MSH receptor in a mouse melanoma cell line. J Recept Signal Transduct Res 1995;15(1-4):43-53.
- Eberle AN. Transformation of an irreversible MSH antagonist into an irreversible MSH agonist by differential receptor crosslinking using the photo-affinity technique. J Mol Recognit 1995;8(1-2):47-51.
- Drozdz R, Chluba-de Tapia J, Eberle AN. [D-Bpa13, Tyr19]MCH, a potent photoreactive analogue of melanin-concentrating hormone for photocrosslinking of MCH receptors. In: Peptides 1994, H.L.S. Maia (ed.), 787-788, ESCOM, Leiden, 1995.
- Drozdz R, Baker BI, Eberle AN. A new radioligand of human/rat melanin concentrating hormone (MCH) for receptor identification. In: Peptides 1994, H.L.S. Maia (ed.), 785-786, ESCOM, Leiden, 1995.
- Siegrist W, Stutz Sibylla, Eberle AN. Regulation of melanotropin receptors in meanoma cells. Extended abstract. J Mol Recognit 1995;8:167-168.
1994
- Dietrich JB, Hildebrand P, Jeker LB, Pansky A, Eberle AN, Beglinger C. Effects of BIM26226, a potent and specific bombesin receptor antagonist, on amylase release and binding of bombesin-like peptides to AR4-2J cells. Regul Pept 1994;53(3):165-173.
- Siegrist W, Stutz S, Eberle AN. Homologous and heterologous regulation of alpha-melanocyte-stimulating hormone receptors in human and mouse melanoma cell lines. Cancer Res 1994;54(10):2604-2610.
1993
- Drozdz R, Baker BI, Zeller A, Eberle AN. Synthesis and biological activity of highly tritiated rat/human melanin concentrating hormone. In: Peptides 1992, CH Schneider, AN Eberle (eds.), 187-188, ESCOM Science Publishers B.V. 1993.
- De Luca M, Siegrist W, Bondanza S, Mathor M, Cancedda R, Eberle AN. Alpha melanocyte stimulating hormone (alpha MSH) stimulates normal human melanocyte growth by binding to high-affinity receptors. J Cell Sci 1993;105 (Pt 4):1079-1084.
- Eberle AN. D1 dopamine receptor mRNA in B16 mouse melanoma cells. Ann N Y Acad Sci 1993;680:660-662.
- Drozdz R, Baker BI, Zeller A, Eberle AN. Synthesis and biological activity of highly tritiated rat/human melanin-concentrating hormone. Ann N Y Acad Sci 1993;680:489-492.
- Lichtensteiger W, Hanimann B, Schlumpf M, Siegrist W, Eberle AN. Pre- and postnatal ontogeny of [125I]Nle4,D-Phe7-alpha-MSH binding sites in rat brain. Ann N Y Acad Sci 1993;680:652-654.
- Bagutti C, Stolz B, Albert R, Bruns C, Pless J, Eberle AN. [111In]DTPA-labeled analogues of alpha-MSH for the detection of MSH receptors in vitro and in vivo. Ann N Y Acad Sci 1993;680:445-447.
- Eberle AN, Siegrist W, Bagutti C, Chluba-De Tapia J, Solca F, Wikberg JE, Chhajlani V. Receptors for melanocyte-stimulating hormone on melanoma cells. Ann N Y Acad Sci 1993;680:320-341.
- Solca FF, Chluba-de Tapia J, Iwata K, Eberle AN. B16-G4F mouse melanoma cells: an MSH receptor-deficient cell clone. FEBS Lett 1993;322(2):177-180.
- Baumann JB, Christen E, Gamboni G, Joss U, van Oostrum J, Girard J, Eberle AN. Receptor binding and biological activity of IL-1 alpha, IL-1 beta, IL-1 beta analogues and an IL-1 antagonist in A375 human melanoma cells. J Recept Res 1993;13(1-4):245-262.
- Eberle AN. Peptides containing multiple photolabels: a new tool for the analysis of ligand-receptor interactions. Reversible long-lasting stimulation and inhibition of MSH receptors by multiple photocrosslinks with alpha-MSH. J Recept Res 1993;13(1-4):27-37.
- Siegrist W, Eberle AN. Homologous regulation of the MSH receptor in melanoma cells. J Recept Res 1993;13(1-4):263-281.
- Bagutti C, Eberle AN. Synthesis and biological properties of a biotinylated derivative of ACTH1-17 for MSH receptor studies. J Recept Res 1993;13(1-4):229-244.
1992
- Siegrist W, Bagutti C, Solca F, Girard J, Eberle AN. MSH receptors on mouse and human melanoma cells: receptor identification, analysis and quantification. Prog Histochem Cytochem 1992;26(1-4):110-118.
- Eberle AN, Siegrist W, Drozdz R, Jäggin Verin V, Bagutti C, Solcà F, Girard J, Zeller A. Radiolabelled melanotropic peptides (α-MSH and MCH) for receptor identification. In: Synthesis and Applications of Isotopically Labelled Compounds 1991, E. Buncel, G.W. Kabalka (eds.), 110-115, Elsevier Science Publishers B.V., 1992.
1991
- Solcà FF, Salomon Y, Eberle AN. Heterogeneity of the MSH receptor among B16 murine melanoma subclones. J Recept Res 1991;11(1-4):379-390.
- Siegrist W, Girard J, Eberle AN. Quantification of MSH receptors on mouse melanoma tissue by receptor autoradiography. J Recept Res 1991;11(1-4):323-331.
- Eberle AN, Verin VJ, Solca F, Siegrist W, Küenlin C, Bagutti C, Stutz S, Girard J. Biologically active monoiodinated alpha-MSH derivatives for receptor binding studies using human melanoma cells. J Recept Res 1991;11(1-4):311-322.
- Eberle AN, Huber M. Antisense peptides: tools for receptor isolation? Lack of antisense MSH and ACTH to interact with their sense peptides and to induce receptor-specific antibodies. J Recept Res 1991;11(1-4):13-43.
- Eberle AN. New perspectives for \’natural\’ therapeutic agents? Karger Gazette 52, 1-4, 1991
- Eberle AN. Peptides – From research tools to \’soft\’ drugs? [1] Chimia 45:145-153, 1991.
- Eberle AN, Huber M. 10. Antisense peptides of ACTH and MSH: tools for receptor isolation? AntNuclAcidProt 1991:187-203.
- Eberle AN, Drozdz R, Solca F, Girard J. Peptides containing multiple photolabels for studies of hormone-receptor interactions. In: Peptides 1990, E. Giralt, D. Andreu (eds.), 692-694, ESCOM Science Publishers B.V., 1991.
1990
- Bird DJ, Baker BI, Eberle AN, Swann RW. The biosynthesis of melanin-concentrating hormone in a fish. J Neuroendocrinol 1990;2:309-315.
- Eberle AN. Gentechnologie und Proteinchemie: Eckpfeiler der modernen Medizin. Mta 1990;5(11):1088-1093.
1989
- Siegrist W, Solca F, Stutz S, Giuffrè L, Carrel S, Girard J, Eberle AN. Characterization of receptors for alpha-melanocyte-stimulating hormone on human melanoma cells. Cancer Res 1989;49(22):6352-6358.
- Solca F, Siegrist W, Drozdz R, Girard J, Eberle AN. The receptor for alpha-melanotropin of mouse and human melanoma cells. Application of a potent alpha-melanotropin photoaffinity label. J Biol Chem 1989;264(24):14277-14281.
- Eberle AN. Gezielte Krebstherapie mit Immunotoxinen und rezeptorgerichteten Toxinpharmaka? Schweiz Rundsch Med Prax 1989;78(18):513-514.
- Kishida M, Baker BI, Eberle AN. The measurement of melanin-concentrating hormone in trout blood. Gen Comp Endocrinol 1989;74(2):221-229.
- Eberle AN, Drozdz R, Baumann JB, Girard J. Receptor-specific antibodies by immunization with \”antisense\” peptides? Pept Res 1989;2(3):213-220.
- Vallarino M, Andersen AC, Delbende C, Ottonello I, Eberle AN, Vaudry H. Melanin-concentrating hormone (MCH) immunoreactivity in the brain and pituitary of the dogfish Scyliorhinus canicula. Colocalization with alpha-melanocyte-stimulating hormone (alpha-MSH) in hypothalamic neurons. Peptides 1989;10(2):375-382.
- Eberle AN, Baker BI, Kishida M, Baumann JB, Girard J. Melanin concentrating hormone. IV. Development of a sensitive solid-phase radioimmunoassay for melanin-concentrating hormone. Life Sci 1989; 45(13):1149-1154.
- Eberle AN, de Graan PN, Scimonelli T, Solca F. Photoaffinity labeling of melanocyte-stimulating hormone receptors. Pharmacol Ther 1989;44(1):63-83.
- Book Review: The melanotropins: chemistry, physiology and mechanism of action. Gen Comp Endocrinol 1989;73:164.
- Eberle AN, Drozdz R, Siegrist W, Baumann JB, Girard J. Synthesis of human \’anti-sense\’ ACTH (\’HTCA\’) and its biological effects. In: Peptides 1988, G. Jung, E. Bayer (eds.), 673-676, Walter de Gruyter, Berlin, New York 1989.
1988
- Girard J, Landolt AM, Valavanis A, Eberle AN, Pampalone A. Results of ACTH and b-LPH determinations in the blood of the inferior petrosal sinus. Adv Biosci 1988;69:353-359.
- Girard J, Zumsteg U, Erb T, Räfle G, Haab G, Pampalone A, Eberle AN, Rochiccioli P, Tauber T. Urinary growth hormone II. Clinical application. Acta Paedriatr. Jpn. 1988;30(suppl.): 205-208.
- Girard J, Zumsteg U, Erb T, Räfle G, Haab G, Pampalone A, Eberle AN, Rochiccioli P, Tauber T. Urinary growth hormone I. Growth hormone excretion in 24 h or timed urine samples reflects plasma growth hormone levels. Acta Paedriatr Jpn 1988;30(suppl.): 201-204.
- Girard J, Landolt AM, Valavanis A, Eberle AN, Pampalone A, Haab G, Jäggin V, Zumsteg U, Zachmann M. Cushing\’s disease: localization of the ACTH-source by ACTH/LPH assays during simultaneous catheterization of left and right sinus petrosus and stimulation with CRH. Acta Paedriatr Jpn 1988;30(suppl.): 244-246.
- Schoofs L, Jegou S, Andersen AC, Tonon MC, Eberle AN, Huybrechts R, De Loof A, Vaudry H. Coexistence of melanin-concentrating hormone and alpha-melanocyte-stimulating hormone immunoreactivities in the central nervous system of the locust, Locusta migratoria. Brain Res 1988;450(1-2):202-208.
- Erb T, Karolyi G, Pampalone A, Eberle AN, Baumann JB, Bürgisser E, Girard J. Human growth hormone in urine: development of an ultrasensitive radiometric assay. Experientia 1988;44(2):155-157.
- Siegrist W, Oestreicher M, Stutz S, Girard J, Eberle AN. Radioreceptor assay for alpha-MSH using mouse B16 melanoma cells+. J Recept Res 1988;8(1-4):323-343.
- Siegrist W, Stutz S, Girard J, Eberle AN. Binding assay for the study of melanoma cell MSH receptors. In: Progress in Cancer Research and Therapy, Vol. 35: Hormones and cancer 3, F. Bresciani, R.J.B. King, M.E. Lippman, J.-P. Raynaud (eds.), 314-317, Raven Press Ltd., New York, 1988.
- Eberle AN, de Graan PNE, Siegrist W, Girard J. Melanotropin receptors: studies with labeled melanotropins. In: Melanotropic peptides Vol. 3(8), 111-127, 1988.
- De Graan PNE, Eberle AN. The role of protein phosphorylation in the mechanism of action of α-MSH. In: Melanotropic peptides Vol. 3(3), 27-44, 1988.
1987
- Scimonelli T, Eberle AN. Photoaffinity labelling of melanoma cell MSH receptors. FEBS Lett 1987;226(1):134-138.
- Pelletier G, Guy J, Désy L, Li S, Eberle AN, Vaudry H. Melanin-concentrating hormone (MCH) is colocalized with alpha-melanocyte-stimulating hormone (alpha-MSH) in the rat but not in the human hypothalamus. Brain Res 1987;423(1-2):247-253.
- Lucas A, Shuster S, Thody AJ, Eberle AN, Girard J. A comparison of structure-activity relationships within alpha-MSH on melanophores of Anolis carolinensis and Rana pipiens. Regul Pept 1987;18(1):43-50.
- De Graan PN, Brussaard AB, Gamboni G, Girard J, Eberle AN. alpha-MSH-induced changes in protein phosphorylation of Cloudman S91 mouse melanoma cells. Mol Cell Endocrinol 1987;51(1-2):87-93.
- Andersen AC, Jegou S, Eberle AN, Tonon MC, Pelletier G, Vaudry H. Coexistence of melanin-concentrating hormone (MCH) and alpha-melanocyte-stimulating hormone (alpha-MSH) in the preoptic nucleus of the frog brain. Brain Res Bull 1987;18(2):257-259.
- Barber LD, Baker BI, Penny JC, Eberle AN. Melanin concentrating hormone inhibits the release of alpha MSH from teleost pituitary glands. Gen Comp Endocrinol 1987;65(1):79-86.
- Scimonelli T, Celis ME, Eberle AN. Changes in alpha-melanocyte-stimulating hormone content in discrete hypothalamic areas of the male rat during a twenty-four-hour period. Horm Res 1987;27(2):78-83.
- Eberle AN, Siegrist W, de Graan PNE, Brussaard AB, Baumann JB, Girard J, Oberholzer MJ, Heitz PU. MSH receptors on mouse melanoma cells: structure-activity studies, receptor labeling and mechanism of signal transduction. In: Cutaneous Melanoma, 217-222, 1987.
1986
- Eberle AN, Atherton E, Dryland A, Sheppard RC. Peptide synthesis. Part 9. Solid-phase synthesis of melanin concentrating hormone using a continuous-flow polyamide method. J Chem Soc Perkin Trans 1986;1:361-367.
- Siegrist W, Eberle AN. In situ melanin assay for MSH using mouse B16 melanoma cells in culture. Anal Biochem 1986;159(1):191-197.
- Andersen AC, Pelletier G, Eberle AN, Leroux P, Jegou S, Vaudry H. Localization of melanin-concentrating hormone-like immunoreactivity in the brain and pituitary of the frog Rana ridibunda. Peptides 1986;7(6):941-951.
- Baumann JB, Eberle AN, Christen E, Ruch W, Girard J. Steroidogenic activity of highly potent melanotropic peptides in the adrenal cortex of the rat. Acta Endocrinol 1986;113(3):396-402.
- Monnet-Tschudi F, Eberle AN, Honegger P. In vivo and in vitro development of alpha-MSH and ACTH in the embryonic and postnatal rat brain. Brain Res 1986;391(1):125-132.
- De Graan PN, Spruijt BM, Eberle AN, Girard J, Gispen WH. ACTH1-4 potentiates alpha-MSH-induced melanophore dispersion and excessive grooming. Peptides 1986;7(1):1-4.
1985
- Eberle AN, Zeller A. Tritiation of peptides to high specific radioactivity. Part 1. Synthesis and biological properties of [13-(3H4)norvaline]-a-MSH and of [2,23-bis-(3H2)tyro-sine]-ACTH(1-24). Helv Chim Acta 1985;68:1880-1892.
- Eberle AN, de Graan PNE. General principles for photoaffinity labeling of peptide hormone receptors. Methods Enzymol 1985;109:129-156.
- Baker BI, Eberle AN, Baumann JB, Siegrist W, Girard J. Effect of melanin concentrating hormone on pigment and adrenal cells in vitro. Peptides 1985;6(6):1125-1130.
- Spruijt BM, De Graan PN, Eberle AN, Gispen WH. Comparison of structural requirements of alpha-MSH and ACTH for inducing excessive grooming and pigment dispersion. Peptides 1985;6(6):1185-1189.
- Eberle AN, Girard J. An Anolis skin melanophore assay suitable for photoaffinity labeling studies with alpha-MSH. Experientia 1985;41(5):654-656.
- Baumann JB, Girard J, Christen E, Eberle AN, Ruch W. Inhibition of the ACTH adrenal response to stress by treatment with hydrocortisone, prednisolone and dexamethasone in the rat. Horm Res 1985;21(4):254-260.
- Eberle AN, Girard J. Photoaffinity labelling of MSH receptors on Anolis melanophores: effects of catecholamines, calcium and forskolin. J Recept Res 1985;5(1):59-81.
- Girard J, Eberle AN. Plasma-ACTH-Bestimmungen für die Differential-Diagnose des Cushing-Syndromes. In: Erkrankungen der Nebenschilddrüsen und Nebennieren, D. Hauri, O. Schmucki (eds.), 162-174, Gustav Fischer Verlag, Stuttgart, 1985.
- Eberle AN, de Graan PNE, Baumann JB, Girard J, van Hees G, van de Veerdonk FCG. Structural requirements of α-MSH for the stimulation of MSH receptors on different pigment cells. In: Pigment Cell 1985. Biological, molecular and clinical aspects of pigmentation. J. Bagnara, S.N. Klaus, E. Paul, M. Schartl (eds.), 191-196, University of Tokyo Press, 1985.
- Eberle AN, Neubert K, Girard J. Tritiation of melanin concentrating hormone to high specific activity: synthesis of (3H4)-norvaline3,6-MCH. In: Peptides: structure and function, C.M. Deber, V.J. Hruby, K.D. Kopple (eds.), 667-670, Pierce Chemical Company, Rockford I11., 1985.
- Eberle AN. Peptide hormone receptors and mechanisms of hormone-receptor interaction. GSIA Pharmacology Course 1985.
- Eberle AN. Receptors for hypophysial hormones: pro-opiomelanocortin and tis peptides (ACTH, MSH, LPH, endorphin). GISA Pharmacology Course 1985.
1984
- Eberle AN. Photoaffinity labelling of MSH receptors on Anolis melanophores: irradiation technique and MSH photolabels for irreversible stimulation. J Receptor Res 1984;4:315-329.
- Walker JE, Gay NJ, Saraste M, Eberle AN. DNA sequence around the Escherichia coli unc operon. Completion of the sequence of a 17 kilobase segment containing asnA, oriC, unc, glmS and phoS. Biochem J 1984;224(3):799-815.
- Eberle AN, de Graan PNE, Girard J. Nitrene and carbene generating photolabels for photoaffinity labeling of MSH receptors on pigment cells. In. Peptides 1984, U. Ragnarsson (ed.), 391-395, Almquist & Wiskell, Stockholm, 1984.
- Girard J, Eberle AN. Stresshormone und frühe Pubertät. Basler Zeitung 1984;51:47.
1983
- Schlegel W, Vecsey A, Eberle AN, Chrétien M, Seidah NG, Zahnd GR. Peptides of the neurointermediate lobe of rat pituitary stimulate growth hormone secretion in vitro. Mol Cell Endocrinol 1983;32:47-55.
- Eberle AN. Photoaffinity labelling of peptide hormone receptors. J Recept Res 1983;3(1-2):313-326.
- Eberle AN, Girad J. Photoreactive [Leu9]-α-MSH derivatives for receptor labeling. In: Peptides 1982, K. Bláha, P. Maloñ (eds.), 589-592, Walter de Gruyter & Co., Berlin, New York 1983.
- Eberle AN. Hormonelle Steuerung der Melanogenese. Hautarzt 1983;34(6):217-219.
1982
- de Graan PN, Eberle AN, van de Veerdonk FC. Calcium sites in MSH stimulation of xenopus melanophores: studies with photoreactive alpha-MSH. Mol Cell Endocrinol 1982;26(3):327-329.
- Walker JE, Eberle AN, Gay NJ, Runswick MJ, Saraste M. Conservation of structure in proton-translocating ATPases of Escherichia coli and mitochondria. Biochem Soc Trans 1982;10:203-206.
- Eberle AN, de Graan PNE, van de Veerdonk FCG. Photoaffinity labeling of MSH receptots with [Apac-Ser1]-α-MSH and [Pap13]-α-MSH. In: Vasopressin, Corticoliberin and ACTH Related Peptides, 231-238, 1982.
- Eberle AN. MSH receptors. In: Melanocyte-stimulating hormone (MSH) and skin: Proceedings of a symposium held at the BAD investigative group meeting, Cardiff, 24 January 1981. Br J Dermatol 1982;106:111-113.
- Walker JE, Eberle AN, Gay NJ, Hanisch P, Saraste M, Runswick MJ. Analysis of the Escherichia coli ATP-synthase complex by DNA and protein sequencing. In: Methods in protein sequence analysis, M. Elzinga (ed.), 337-354, The Humana Press, 1982.
1981
- Saraste M, Gay NJ, Eberle AN, Runswick MJ, Walker JE. The atp operon: nucleotide sequence of the genes for g, b, and e subunits of Escherichia coli ATP synthase. Nucleic Acids Res 1981;9:5287-5296.
- Eberle AN, de Graan PNE, Hübscher W. Synthesis and biological properties of p-azidophenylalanine13-a-melanotropin, a potent photoaffinity label for MSH receptors. Helv Chim Acta 1981;64:2645-2653.
- Monnet F, Reubi J-C, Eberle AN, Lichtensteiger W. Diurnal variation in the release of a-MSH from rat hypothalamus and pituitary. Neuroendocrinology 1981;33:284-287.
- Schwyzer R, Do KQ, Eberle AN, Fauchère J-L. Synthesis and biological properties of enkephalin-like peptides containing carboranylalanine in place of phenylalanine. Helv Chim Acta 1981;64:2078-2083.
- Kriwaczek VM, Bristow AF, Eberle AN, Gleed C, Schulster D, Schwyzer R. Superpotency and superaffinity phenomena in the stimulation of steroidogenesis in adrenocortical cells by adrenocorticotropin-tobacco mosaic virus conjugates. Mol Cell Biochem 1981;40(1):49-59.
- De Graan PNE, Eberle AN, van de Veerdonk FCG. Photoaffinity labelling of MSH receptors reveals a dual role of calcium in melanophore stimulation. FEBS Lett 1981;129:113-116.
- van Wimersma Greidanus TB, de Rotte GA, Thody AJ, Eberle AN. Melanocyte-stimulating hormone and adaptive behaviour. Ciba Found Symp 1981;81:277-294.
- Eberle AN. Structure and chemistry of the peptide hormones of the intermediate lobe. Ciba Found Symp 1981;81:13-31.
- De Graan PNE, Eberle AN, van de Veerdonk FCG. Photoaffinity labeling of MSH receptors of Xenopus melanophores. In: Pigment Cell 1981. Phenotypic Expression in Pigment Cells. M. Seiji (ed.), 373-379, University of Tokyo Press 1981.
- Eberle AN, Kriwaczek VM, Schulster D. Corticotropin and melanotropin: organization and transmission of hormonal information. In: Perspectives in Peptide Chemistry, A.N. Eberle, R. Geiger, T. Wieland (eds.), 407-422, S. Karger, Basel 1981.
1980
- De Graan PN, Eberle AN. Irreversible stimulation of Xenopus melanophores by photoaffinity labelling with p-azidophenylalanine13-alpha-melanotropin. FEBS Lett 1980;116(1):111-115.
- Eberle AN. MSH receptors. In: Cellular receptors for hormones and neurotransmitters. D. Schulster, A. Levitzki (eds.), 219-231, John Wiley & Sons Ltd. 1980.
- Celio MR, Höllt V, Buetti G, Pasi A, Bürgisser E, Eberle AN, Kopp G, Siebenmann R, Friede RL, Landolt A, Binz H, Zenker W. Immunohistochemical study of beta-endorphin and related peptides in the “invading cells” of the human neurohypophysis during ontogenesis and adulthood. In: Neuronal Peptides and Neuronal Comminication. E. Costa, M. Trabucchi (eds.), 271-283, Raven Press, New York 1980.
- Eberle AN. Studies on melanotropin (MSH) receptors of melanophores and melanoma cells. Biochem Soc Trans 1980;9(1):37-39.
1979
- Eberle AN, Hübscher W. a-Melanotropin labelled at its tyrosine2 residue: synthesis and biological activities of 3′-iodotyrosine2-, 3′-125iodotyrosine2-, 3′,5′-diiodotyrosine2- and (3′,5′-3H2)tyrosine2-a-melanotropin, and of related peptides. Helv Chim Acta 1979;62:2460-2483.
- Eberle AN, Schwyzer R. Divergent melanophore-dispersing and tyrosinase-stimulating activity of synthetic leucine9-a-melanotropin. Helv Chim Acta 1979;62:2452-2459.
- Fauchère J-L, Leukart O, Eberle AN, Schwyzer R. The synthesis of [4-carboranylalanine, 5-leucine]-enkephalin. Helv Chim Acta 1979;62:1385-1395.
- Castell JV, Eberle AN, Kriwaczek VM, Tun-Kyi A, Schiller PW, Do KQ, Thanei P, Schwyzer R. [D-Ala2, Phe(p-NO2)4, Leu5]-Enkephalin amide and Na-[D-Ala2, Leu5]-enkephalyl-Ne-acetyl-lysine amide: synthesis and biological properties of prospective enkephalin cooperative affinity and photoaffinity labels. Helv Chim Acta 1979;62:525-529.
- Zahnd GR, Vecsey A, Eberle AN. Structure-function studies on the growth hormone releasing activity of alpha-melanotropin. Acta Endocr Suppl 225:223, 1979.
- Kriwaczek VM, Eberle AN, Schwyzer R. Tobacco mosaic virus as a carrier for peptide hormones. In: Peptides 1978, I.Z. Siemion (ed.), 597-599, Wroclaw University Press, Poland 1979.
- Eberle AN, Schwyzer R. Synthesis of specifically labeled alpha-melanotropin derivatives. In: Peptides 1978, I.Z. Siemion (ed.), 589-592, Wroclaw University Press, Poland 1979.
- Eberle AN, Kriwaczek VM, Schwyzer R. Studies on tyrosinase stimulation, binding and degradation of alpha-MSH interacting with non-synchronized mouse melanoma cells in culture. In: Peptides: Structure and Biological Function, E. Gross, J. Meienhofer (eds.), 1033-1036, Pierce Chemical Company 1979.
- Schwyzer R, Eberle AN, Kriwaczek VM. Studies on the use of carboranylalanine for neutron activation therapy (234). Curr Cancer Res 1979;35.
- Eberle AN, Schwyzer R. Mutiply labeled alpha-MSH derivatives for degradation studies. Experientia 1979;35:911.
1978
- Eberle AN, Chang Y-S, Schwyzer R. Chemical synthesis and biological activity of the dogfish (Squalus acanthias) a-melanotropin I and II, and of related peptides. Helv Chim Acta 1978;61:2360-2374.
- Kriwaczek VM, Eberle AN, Müller M, Schwyzer R. Tobacco mosaic virus as a carrier for small molecules. I. The preparation and characterization of a TMV/a-melanotropin conjugate. Helv Chim Acta 1978;61:1232-1240.
- Eberle AN, Kriwaczek VM, Schwyzer R. Mechanism of alpha-melanotropin action. Bull Schweiz Akad Med Wiss 1978;34:99-111.
- Eberle AN. Aspekte der molekularen Linguistik bei der Informations-übertragung durch Peptidhormone. 2. Frühjahrskolloqium Bremen 30.3.-1.4.1978, “Zelluläre Kommunikations- und Kontrollmechanismen”, 1-15.
1977
- Schwyzer R, Eberle AN. On the molecular mechanism of a-MSH receptor interactions. Front Hormone Res 1977;4:18-25.
- Eberle AN, Hübscher W, Schwyzer R. Synthese von radioaktiv markierten Bromacetyl- und Diazoacetyl-a-melanotropin-Derivaten zum Studium von kovalenten Hormon-Makromolekül-Komplexen. Helv Chim Acta 1977;60:2895-2910.
- Eberle AN, Leukart O, Schiller P, Fauchère J-L, Schwyzer R. Hormone-receptor interactions: [4-carboranylalanine, 5-leucine]-enkephalin as a structural probe for the opiate receptor. FEBS Lett 1977;82:325-328.
- Eberle AN, Kriwaczek VM, Schwyzer R. Hormone-receptor interactions: melanotropic activities of covalent serum albumin complexes with a-melanotropin, a-melanotropin fragments, and enkephalin. FEBS Lett 1977; 80:246-250.
- Kopp HG, Eberle AN, Vitins P, Lichtensteiger W, Schwyzer R. Specific antibodies against a-melanotropin for radioimmunoassay. Eur J Biochem 1977;75:417-422.
- Schwyzer R et al. 1. Anterior pituitary hormones. In: Amino Acids Peptides and Proteins. Chemical structure and biological activity of hormones and related compounds. 1977;5:405-418.
- Kriwaczek VM, Eberle AN, Vollenweider HJ, Schwyzer R. Alpha-melanotropin-macromolecule complexes. Experentia 1977;33.
1976
- Eberle AN, Schwyzer R. Synthese von [D-Alanin1, 4’azido-3′,5′-ditritio-L-phenylalanin2, norvalin4]-a-melanotropin als “Photoaffinitätsprobe” für Hormon-Rezeptor-Wechselwirkungen. Helv Chim Acta 1976;59:2421-2431.
- Leukart O, Caviezel M, Eberle AN, Escher E, Tun-Kyi A, Schwyzer R. L-o-Carboranylalanine, a boron-analogue of phenylalanine. Helv Chim Acta 1976;59:2184-2187.
- Leukart O, Caviezel M, Eberle AN, Escher E, Tun-Kyi A, Schwyzer R. Synthesis of L-propargylglycine and derivatives. Helv Chim Acta 1976;59:2181-2183.
- Fischli W, Caviezel M, Eberle AN, Escher E, Schwyzer R. Synthese von 4′-Azido-3′,5′-ditritio-L-phenylalanin-peptiden als “Photoaffinitätsproben” für Ligand-Rezeptor-Wechselwirkungen. Helv Chim Acta 1976;59:878-879.
- Eberle AN, Schwyzer R. Hormone-receptor interactions. The message sequence of a-melanotropin: demonstration of two active sites. Clin Endocrinol 1976;5:41s-48s.
- Eberle AN, Schwyzer R. Alpha-melanotropin receptors: non-identical hormonal message sequences (active sites) triggering receptors in melanocytes, adipocytes and CNS cells. In: Surface Membrane Receptors. R.A. Bradshaw, W.A. Frazier, R.C. Merrell, D.I. Gottlieb, R.A. Hogue-Angeletti (eds.), 291-304, Plenum Publishing Corporation, New York 1976.
1975
- Eberle AN, Fauchère J-L, Tesser GI, Schwyzer R. Hormon-Rezeptor-Wechselwirkungen. Synthese von a-Melanotropin und von informations-tragenden Teilsequenzen unter Verwendung alkalilabiler Schutzgruppen. Helv Chim Acta 1975;58:2106-2129.
- Eberle AN, Schwyzer R. Hormone-receptor interactions. Demonstration of two message sequences (active sites) in a-melanotropins. Helv Chim Acta 1975; 58:1228-1235.
1973
1972